Babban Matsayin Magunguna na Tsabta 1421373-66-1 Mesylate-AZD9291 don Maganin Ciwon daji
Samfurasuna | Saukewa: AZD-9291 |
Makamantu | N-[2-[[2- (Dimethylamino) ethyl] methylamino] -4-methoxy-5-[4- (1-methyl-1H-indol-3-yl) -2-pyrimidinyl] amino] phenyl] - 2-propenamide methanesulfonate (1: 1) |
CAS No. | 1421373-66-1 |
Bayyanar | Fari zuwa haske rawaya m foda |
Tsarin kwayoyin halitta | C28H33N7O2CH4O3S |
Nauyin Kwayoyin Halitta | 595.71 |
Amfani | Matsayin Magunguna ko Manufar Bincike |
Shiryawa | Kamar yadda kuka bukata |
Adana | Ajiye a cikin matsi, kwantena masu jure haske a wuri mai sanyi |
Saukewa: AZD-9291Saukewa: 1421373-66-1 | ||
Iabubuwa | Standards | Rsakamakon |
Bayyanar | Fari zuwa haske rawaya m foda | Hasken rawaya m foda |
Ihakora | By IR | Ya bi |
Farashin HPLC | Ya bi | |
Solubility | Mai narkewa a cikin Dimethylsulfoxide, dan kadan mai narkewa a cikin Ethanol da Acetonitrile, tare da narkar da ruwa mai dogaro da pH. | Ya bi |
Abubuwan Ruwa (KF) | ≤ 1.00% | 0.42% |
Ragowa akan Ignition | 0.10% | 0.05% |
HsaukiMetal | ≤ 20pm | Ya bi |
Mesylate | 15.20% ~ 18.20% | 15.90% |
Ragowar Magani | Acetonitrile: ≤410ppm | ND |
Acetone: ≤5000ppm | ND | |
Tetrahydrofuran: ≤720ppm | ND | |
RmurnaSabubuwa | Matsakaicin ƙazanta ɗaya: ≤0.20% | 0.17% |
Jimlar ƙazanta: ≤1.00% | 0.25% | |
Girman Barbashi | D90: ≤100μm | 57.97% |
Ace (HPLC bisa bushewa) | 98.00% ~ 102.00% | 99.80% |
Matsayin Magana | In-gida Standard |
Bayanin Kamfanin
√ Cikakken ƙwarewar gudanarwa a masana'anta da ƙwararrun masu bin fasaha; √ Quality ne ko da yaushe mu saman la'akari, M QC tsarin; √ 11 shekaru gogaggen fitar da tallace-tallace tawagar; √ R&D mai zaman kansa; √ Biyu da aka sanya hannu na dogon lokaci na GMP; √ wadataccen albarkatu na masana'antu marasa aiki da yawa don aikin da aka keɓance; √ Ƙwararren aiki mai inganci tare da madaidaiciyar hanya.Ku rubuta sakonku anan ku aiko mana